Deschloroetizolam

Deschloroetizolam (also known as Etizolam-2) is a thienotriazolodiazepine that is the dechlorinated analog of the closely related etizolam.[1][2][3] The compound has been sold as a designer drug.[4][5][6]

Deschloroetizolam

Clinical data
Dependence liability	Moderate
Routes of administration	Oral, sublingual, rectal
Legal status
Legal status	CA: Schedule IV DE: NpSG (Industrial and scientific use only) UK: Under Psychoactive Substances Act Illegal in Sweden
Identifiers
IUPAC name 4-phenyl-2-ethyl-9-methyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepine
CAS Number	40054-73-7
PubChem CID	827322
ChemSpider	722596
UNII	69HF7J354D
Chemical and physical data
Formula	C17H16N4S
Molar mass	308.40 g·mol^−1
3D model (JSmol)	Interactive image
SMILES CCC1=CC2=C(S1)N3C(=NN=C3CN=C2C4=CC=CC=C4)C
InChI InChI=1S/C17H16N4S/c1-3-13-9-14-16(12-7-5-4-6-8-12)18-10-15-20-19-11(2)21(15)17(14)22-13/h4-9H,3,10H2,1-2H3 Key:JIOBORXCOGMHSV-UHFFFAOYSA-N

Legal status

Deschloroetizolam is classified and controlled as a hazardous substance in Sweden as of on October 15, 2015.[7]

See also

• Adinazolam
• Clonazolam
• Diclazepam
• Etizolam
• Flubromazepam
• Flubromazolam
• Meclonazepam
• Metizolam
• Nifoxipam
• Pyrazolam

References

1. Weber KH, Bauer A, Langbein A, Daniel H (September 1978). "Heteroaromaten mit anellierten Siebenringen, III. Umwandlung von Thienotriazolooxazepinen in Diazepine". Justus Liebigs Annalen der Chemie (in German). 1978 (8): 1257–1265. doi:10.1002/jlac.197819780806.
2. US 3904641, Nakanishi M, Tahara T, Araki K, Shiroki M, "Triazolothienodiazepine compounds", assigned to Yoshitomi Pharmaceutical Industries, Ltd.
3. EP 0776892, Hiroshi K, Syuji E, Hideaki S, Minoru M, Kenichi O, "Thienylazole compound and thienotriazolodiazepine compound", published 4 June 1997, assigned to Yoshitomi Pharmaceutical Industries, Ltd.
4. "Deschloroetizolam". New Synthetic Drugs Database.
5. Pettersson Bergstrand M, Helander A, Hansson T, Beck O (April 2017). "Detectability of designer benzodiazepines in CEDIA, EMIT II Plus, HEIA, and KIMS II immunochemical screening assays". Drug Testing and Analysis. 9 (4): 640–645. doi:10.1002/dta.2003. PMID 27366870.
6. Manchester KR, Maskell PD, Waters L (March 2018). "a and plasma protein binding values for benzodiazepines appearing as new psychoactive substances" (PDF). Drug Testing and Analysis. 10 (8): 1258–1269. doi:10.1002/dta.2387. PMID 29582576.
7. "Nya substanser klassas som narkotika eller hälsofarlig vara" (in Swedish). Folkhälsomyndigheten. 18 August 2015.